| US 7,572,818 B2 | ||
| 2-pyridylethylbenzamide derivative | ||
| Darren James Mansfield, Lyons (France); Tracey Cooke, St Albans (United Kingdom); Peter Stanley Thomas, Cambridge (United Kingdom); Pierre-Yves Coqueron, Lyons (France); Jean-Pierre Vors, Lyons (France); Geoffrey Gower Briggs, Herts (United Kingdom); Hélène Lachaise, Lyons (France); Heiko Rieck, Sainte Foy les Lyons (France); Philippe Desbordes, Lyons (France); and Marie-Claire Grosjean-Cournoyer, Curis Au Mont d'Or (France) | ||
| Assigned to Bayer Cropscience S.A., (France) | ||
| Appl. No. 10/524,345 PCT Filed Aug. 08, 2003, PCT No. PCT/EP03/09516 § 371(c)(1), (2), (4) Date Feb. 11, 2005, PCT Pub. No. WO2004/016088, PCT Pub. Date Feb. 26, 2004. |
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| Claims priority of application No. 02356159 (EP), filed on Aug. 12, 2002; and application No. 03 05233 (FR), filed on Apr. 29, 2003. | ||
| Prior Publication US 2005/0234110 A1, Oct. 20, 2005 | ||
| Int. Cl. A61K 31/44 (2006.01) | ||
| U.S. Cl. 514—357 [546/337] | 16 Claims |
1. A compound of the general formula (I):
 p is an integer equal to 1, 2, 3 or 4;
q is an integer equal to 1, 2, 3, 4 or 5;
each X is independently selected from the group consisting of halogen, alkyl, and haloalkyl, provided that at least one X
is a haloalkyl;
each Y is independently selected from the group consisting of halogen, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, amino,
phenoxy, alkylthio, dialkylamino, acyl, cyano, ester, hydroxyl, aminoalkyl, benzyl, haloalkoxy, halosulphonyl, halothioalkyl,
alkoxyalkenyl, alkylsulphonamide, nitro, alkylsulphonyl, phenylsulphonyl, and benzylsulphonyl;
as to the N-oxides of 2-pyridine thereof;
with the exception of N-{2-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]ethyl}-2,6 -dichlorobenzamide.
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